Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of kd for PROTEIN FARNESYLTRANSFERASE/GERANYLGERANYLTRANSFERASE TYPE-1 SUBUNIT ALPHA
having polymerids = 1377,1381,1383,50001266 and
complexids = 50000153,50000414,162,164,50000105,50000155,50003567,160,163,50000022,5000007...
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50366477(CHEMBL69330)
Affinity DataKd:  75nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50559445(CHEMBL4758112)
Affinity DataKd:  340nMAssay Description:Displacement of (1-(2-aminoethyl)-3,5-dimethyl-1H-pyrazol-4-yl)(4-((1-neopentyl-1H-benzo[d]imidazol-2-yl)methyl)piperazin-1-yl)methanone from FNTA in...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50366477(CHEMBL69330)
Affinity DataKd:  2nMAssay Description:Binding affinity to FTase (unknown origin)More data for this Ligand-Target Pair